US 12,145,902 B2
Solid presentation form of at least one phenol derivative and process for obtaining same
Rodolphe Sapey-Triomphe, Sérézin-du-Rhône (FR); and Cédric Humblot, Lyons (FR)
Assigned to SPECIALTY OPERATIONS FRANCE, Lyons (FR)
Appl. No. 17/266,238
Filed by SPECIALTY OPERATIONS FRANCE, Lyons (FR)
PCT Filed Aug. 2, 2019, PCT No. PCT/EP2019/070872
§ 371(c)(1), (2) Date Feb. 5, 2021,
PCT Pub. No. WO2020/030541, PCT Pub. Date Feb. 13, 2020.
Claims priority of application No. 1857419 (FR), filed on Aug. 9, 2018.
Prior Publication US 2021/0292262 A1, Sep. 23, 2021
Int. Cl. A61K 8/02 (2006.01); A23L 27/20 (2016.01); A61K 9/20 (2006.01); C07C 41/40 (2006.01); C07C 43/23 (2006.01)
CPC C07C 43/23 (2013.01) [A23L 27/204 (2016.08); A61K 8/0216 (2013.01); A61K 9/2072 (2013.01); C07C 41/40 (2013.01); A23V 2002/00 (2013.01); C07C 2601/16 (2017.05)] 20 Claims
OG exemplary drawing
 
1. A novel solid presentation form comprising at least one rounded part; a pellet; or a spherical cap; wherein the novel solid presentation form, pellet, or spherical cap comprises at least one compound of formula (I)

OG Complex Work Unit Chemistry
wherein:
n is between 0 and 5,
R1 is selected from the group consisting of hydrogen, alkyl, and alkenyl,
R2 is selected from the group consisting of hydroxyl, alkyl, alkenyl, alkynyl, alkoxy, formyl, and acetyl, and
the novel presentation form, the pellet, and the spherical cap each comprise at least one flat part that is a continuous surface and represents at least 5% of the total surface of each of the novel presentation form, the pellet and the spherical cap.