US 12,139,497 B2
Aryl, heteroaryl, and heterocyclic compounds for treatment of medical disorders
Jason Allan Wiles, Madison, CT (US); Avinash S. Phadke, Branford, CT (US); Milind Deshpande, Madison, CT (US); Atul Agarwal, Hamden, CT (US); Dawei Chen, Guilford, CT (US); Venkat Rao Gadhachanda, Hamden, CT (US); Akihiro Hashimoto, Branford, CT (US); Godwin Pais, Hamden, CT (US); Qiuping Wang, Bethany, CT (US); and Xiangzhu Wang, Branford, CT (US)
Assigned to Achillion Pharmaceuticals, Inc., Boston, MA (US)
Filed by Achillion Pharmaceuticals, Inc., Boston, MA (US)
Filed on Mar. 21, 2023, as Appl. No. 18/124,427.
Application 18/124,427 is a division of application No. 17/015,171, filed on Sep. 9, 2020, abandoned.
Application 16/351,203 is a division of application No. 16/010,081, filed on Jun. 15, 2018, granted, now 10,287,301, issued on May 14, 2019.
Application 17/015,171 is a continuation of application No. 16/351,203, filed on Mar. 12, 2019, granted, now 10,822,352, issued on Nov. 3, 2020.
Application 16/010,081 is a continuation of application No. 15/247,399, filed on Aug. 25, 2016, granted, now 10,011,612, issued on Jul. 3, 2018.
Claims priority of provisional application 62/209,972, filed on Aug. 26, 2015.
Prior Publication US 2023/0287005 A1, Sep. 14, 2023
Int. Cl. C07D 513/04 (2006.01); A61K 31/167 (2006.01); A61K 31/395 (2006.01); A61K 31/40 (2006.01); A61K 31/416 (2006.01); A61K 31/4439 (2006.01); A61K 31/444 (2006.01); A61K 31/497 (2006.01); A61K 31/506 (2006.01); A61K 31/519 (2006.01); A61K 38/00 (2006.01); A61P 1/16 (2006.01); A61P 3/06 (2006.01); A61P 9/00 (2006.01); A61P 9/10 (2006.01); A61P 11/00 (2006.01); A61P 13/00 (2006.01); A61P 13/02 (2006.01); A61P 17/00 (2006.01); A61P 19/02 (2006.01); A61P 21/00 (2006.01); A61P 25/00 (2006.01); A61P 25/02 (2006.01); A61P 27/00 (2006.01); A61P 27/02 (2006.01); A61P 29/00 (2006.01); A61P 37/02 (2006.01); A61P 43/00 (2006.01); C07D 401/14 (2006.01); C07D 403/06 (2006.01); C07D 403/14 (2006.01); C07D 405/14 (2006.01); C07D 409/14 (2006.01); C07D 413/14 (2006.01); C07D 417/04 (2006.01); C07D 417/14 (2006.01); C07D 471/04 (2006.01); C07D 487/04 (2006.01); C07D 493/04 (2006.01); C07D 495/04 (2006.01)
CPC C07D 513/04 (2013.01) [C07D 401/14 (2013.01); C07D 403/06 (2013.01); C07D 403/14 (2013.01); C07D 405/14 (2013.01); C07D 409/14 (2013.01); C07D 413/14 (2013.01); C07D 417/14 (2013.01); C07D 471/04 (2013.01); C07D 487/04 (2013.01); C07D 493/04 (2013.01); C07D 495/04 (2013.01)] 20 Claims
 
1. A compound or a pharmaceutically acceptable salt thereof, wherein the compound is selected from:

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