CPC C07D 471/04 (2013.01) [A61K 45/06 (2013.01)] | 19 Claims |
1. A compound represented by formula (I):
A-B—C (I)
wherein:
A is
B is alkylene;
C is
R is H, alkyl, or aryl;
R1 is independently H, alkyl, halide, alkoxy, CF3, OH, NO2, —N(H)R, or NH2;
R2 is H, alkyl, substituted or unsubstituted aryl, substituted or unsubstituted heteroaryl, alkoxy, —OH, N(R)C(O)R4, or —N(R)-heteroaryl;
R3 is independently alkyl, halide, alkoxy, CF3, OH, NO2, or NH2;
R4 is alkyl, cycloalkyl, heterocycloalkyl, aryl, heteroaryl, -alkylene-heterocyclyl, -alkylene-N(R)C(O)R5, or -alkylene-N(R)—SO2Me;
R5 is alkyl, or cycloalkyl;
R6 is H, or alkyl;
X is N;
Rd is H, or (C1-C6)alkyl;
a is independently 0, or 1; and
b is 0, 1, 2, 3, or 4;
or a pharmaceutically acceptable salt thereof.
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