US 12,419,308 B2
Phenylpyrazole insecticide compounds and compositions
Francesco Dottorini, Perugia (IT); Aurora Valeri, Siena (IT); and Alessandra Di Veroli, Perugia (IT)
Assigned to Molecular Horizon SRL, Bettona (IT)
Filed by Molecular Horizon SRL, Bettona (IT)
Filed on Nov. 25, 2024, as Appl. No. 18/959,040.
Application 18/959,040 is a continuation of application No. PCT/EP2024/062844, filed on May 8, 2024.
Claims priority of application No. 23425020 (EP), filed on May 9, 2023.
Prior Publication US 2025/0089719 A1, Mar. 20, 2025
Int. Cl. C07D 471/04 (2006.01); A01N 43/90 (2006.01); A01P 7/02 (2006.01); A61K 9/00 (2006.01); A61K 31/437 (2006.01); A61P 33/14 (2006.01)
CPC A01N 43/90 (2013.01) [A01P 7/02 (2021.08); A61K 9/0017 (2013.01); A61K 31/437 (2013.01); A61P 33/14 (2018.01); C07D 471/04 (2013.01)] 20 Claims
 
1. A compound having the following general structure,

OG Complex Work Unit Chemistry
wherein R1 and R2 are each independently selected from H, halo, cyano, nitro, hydroxy, amino, C1-6alkyl, C3-6cycloalkyl, C1-6haloalkyl, C1-6alkoxy, C1-6haloalkoxy, C3-6cycloalkoxy, C3-6halocycloalkyl, NH(C1-6alkyl), N(C1-6alkyl)(C1-6alkyl), and
3-6 membered heterocycloalkyl; and
each R is independently selected from halo, cyano, nitro, hydroxy, amino, C1-6alkyl,
C3-6cycloalkyl, C1-6haloalkyl, C1-6alkoxy, C1-6haloalkoxy, and C3-6halocycloalkyl;
in free or salt form.