CPC C07K 16/40 (2013.01) [A61B 5/0042 (2013.01); A61B 5/055 (2013.01); A61B 6/032 (2013.01); A61B 6/501 (2013.01); A61P 25/00 (2018.01); C07K 16/18 (2013.01); G01N 33/6896 (2013.01); C07K 2317/20 (2013.01); C07K 2317/21 (2013.01); C07K 2317/34 (2013.01); C07K 2317/52 (2013.01); C07K 2317/565 (2013.01); C07K 2317/76 (2013.01); C07K 2317/92 (2013.01)] | 20 Claims |
1. An antibody or antigen-binding fragment thereof that specifically binds to a human ubiquitin c-terminal hydrolase L1 (UCH-L1) protein, comprising:
a heavy chain variable region that comprises CDR-H1, CDR-H2, and CDR-H3 amino acid sequences; and
a light chain variable region that comprises CDR-L1, CDR-L2, and CDR-L3 amino acid sequences,
wherein:
(1) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:2, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:10, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:21; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:29, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:38, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:46; or
(2) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:5, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:13, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:23; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:32, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:39, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:47; or
(3) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:3, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:11, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:20; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:30, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:37, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:45; or
(4) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:4, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:12, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:22; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:31, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:39, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:47; or
(5) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:6, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:14, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:24; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:33, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:40, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:48; or
(6) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:6, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:14, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:24; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:34, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:41, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:48; or
(7) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:6, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:15, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:24; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:34, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:42, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:48; or
(8) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:6, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:14, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:24; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:35, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:41, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:48; or
(9) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:6, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:16, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:25; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:34, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:42, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:48; or
(10) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:7, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:17, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:26; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:36, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:43, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:49; or
(11) the heavy chain variable region comprises (i) the CDR-H1 amino acid sequence comprising SEQ ID NO:8, (ii) the CDR-H2 amino acid sequence comprising SEQ ID NO:18, and (iii) the CDR-H3 amino acid sequence comprising SEQ ID NO:27; and
the light chain variable region comprises (i) the CDR-L1 amino acid sequence comprising SEQ ID NO:36, (ii) the CDR-L2 amino acid sequence comprising SEQ ID NO:44, and (iii) the CDR-L3 amino acid sequence comprising SEQ ID NO:49.
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