US 12,384,773 B2
Thiazole compounds and methods of use thereof
Srijita Bhowmik, Hayward, CA (US); Karen Yir Jing Chen, Hayward, CA (US); Jenna Leigh Jeffrey, Hayward, CA (US); Manjunath Lamani, Hayward, CA (US); Manmohan Reddy Leleti, Hayward, CA (US); Guillaume Mata, Hayward, CA (US); Hyunyoung Moon, Hayward, CA (US); Pradeep Nareddy, Hayward, CA (US); Srinivas Paladugu, Hayward, CA (US); Zhang Wang, Foster City, CA (US); Xuelei Yan, Hayward, CA (US); Monika Yadav, Hayward, CA (US); and Jiang Zhu, Hayward, CA (US)
Assigned to Arcus Biosciences, Inc., Hayward, CA (US)
Filed by Arcus Biosciences, Inc., Hayward, CA (US)
Filed on Nov. 1, 2024, as Appl. No. 18/934,931.
Claims priority of provisional application 63/563,078, filed on Mar. 8, 2024.
Claims priority of provisional application 63/595,707, filed on Nov. 2, 2023.
Prior Publication US 2025/0145606 A1, May 8, 2025
Int. Cl. C07D 417/12 (2006.01); A61K 31/426 (2006.01); A61K 31/427 (2006.01); A61K 31/429 (2006.01); A61K 31/433 (2006.01); A61K 31/4355 (2006.01); A61K 31/436 (2006.01); A61K 31/4439 (2006.01); A61K 31/496 (2006.01); A61K 31/497 (2006.01); A61K 31/4985 (2006.01); A61K 31/501 (2006.01); A61K 31/506 (2006.01); A61K 31/5377 (2006.01); C07D 277/56 (2006.01); C07D 417/14 (2006.01); C07D 487/04 (2006.01); C07D 491/048 (2006.01); C07D 491/052 (2006.01); C07D 513/04 (2006.01)
CPC C07D 417/12 (2013.01) [A61K 31/426 (2013.01); A61K 31/427 (2013.01); A61K 31/429 (2013.01); A61K 31/433 (2013.01); A61K 31/4355 (2013.01); A61K 31/436 (2013.01); A61K 31/4439 (2013.01); A61K 31/496 (2013.01); A61K 31/497 (2013.01); A61K 31/4985 (2013.01); A61K 31/501 (2013.01); A61K 31/506 (2013.01); A61K 31/5377 (2013.01); C07D 277/56 (2013.01); C07D 417/14 (2013.01); C07D 487/04 (2013.01); C07D 491/048 (2013.01); C07D 491/052 (2013.01); C07D 513/04 (2013.01)] 14 Claims
 
1. A compound selected from the group consisting of

OG Complex Work Unit Chemistry