| CPC C12Q 1/6895 (2013.01) [C07H 21/04 (2013.01); C12Q 1/6844 (2013.01); C12Q 1/6848 (2013.01); C12Q 1/6853 (2013.01); C12Q 1/6876 (2013.01); C12Q 1/689 (2013.01); C12Q 2600/156 (2013.01)] | 10 Claims |
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1. A method of designing a primer oligonucleotide, the primer oligonucleotide comprising from 5′ to 3′:
i) a first region comprising a self-complementary sequence comprising from 5′ to 3′ the reverse complement of a nicking enzyme recognition sequence, a palindromic sequence, and the nicking enzyme recognition sequence, and
ii) a second region at least 16 nucleotides long that specifically binds to a complementary region on a target nucleic acid molecule, wherein the second region of the primer oligonucleotide comprises two or more 2′ modified nucleotides, wherein the two or more 2′ modified nucleotides are selected from the group consisting of 2′-O—methyl, 2′-methoxyethoxy, 2′-fluoro, 2′-hydroxyl, 2′-alkyl, 2′-allyl, 2′-O-[2-(methylamino)-2-oxoethyl], 4′-CH2—O-2′-bridge, 4′-(CH2)2—O-2′-bridge, 2′-LNA, and 2′-O-(N-methylcarbamate) and those comprising base analogs, and wherein two or more 2′ modified nucleotides are contiguous;
the method comprising:
a) selecting the second region of said primer oligonucleotide, so that the ΔG for a double-stranded primer-target hybrid formed by the hybridization of the second region and the target nucleic acid molecule is at least 15 kcal/mol lower than the ΔG of a self-dimer comprising the second region of the primer; and
b) selecting a first region of said primer oligonucleotide, so that the ΔG for a homodimer formed by hybridization of the self-complementary first region of two primer oligonucleotide molecules is at least 15 kcal/mol lower than the ΔG of a self-dimer comprising the second region of the primer oligonucleotide.
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