CPC C07K 5/0808 (2013.01) [A61K 47/6817 (2017.08); C07K 5/0205 (2013.01); C07K 9/003 (2013.01); C07K 16/28 (2013.01); C07K 16/30 (2013.01); C07K 16/40 (2013.01); A61K 38/00 (2013.01); A61K 47/6855 (2017.08); C07K 5/06078 (2013.01); C07K 2317/76 (2013.01)] | 12 Claims |
1. A compound according to Formula 1000:
![]() or a pharmaceutically acceptable salt, solvate, stereoisomer, or tautomer thereof, wherein:
Ar is a divalent six-membered, substituted or unsubstituted, monocyclic aryl; divalent five- or six-membered, substituted or unsubstituted, monocyclic heteroaryl; divalent nine- or ten-membered, substituted or unsubstituted, monocyclic aryl; or a divalent eight-, nine- or ten-membered, substituted or unsubstituted, fused bicyclic aryl or heteroaryl;
L is absent or —CH2—;
X is
![]() R is hydrogen; and
W1, W2, W3, W4, W5, EG, each RT, and HP are all absent, SG is a single bond.
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