US 12,187,686 B2
BRD4-JAK2 inhibitors
Ernst Schönbrunn, Tampa, FL (US); Nicholas J. Lawrence, Tampa, FL (US); Harshani R. Lawrence, Tampa, FL (US); and Gary Reuther, Tampa, FL (US)
Assigned to H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC., Tampa, FL (US)
Appl. No. 17/274,287
Filed by H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC., Tampa, FL (US)
PCT Filed Sep. 9, 2019, PCT No. PCT/US2019/050147
§ 371(c)(1), (2) Date Mar. 8, 2021,
PCT Pub. No. WO2020/051571, PCT Pub. Date Mar. 12, 2020.
Claims priority of provisional application 62/728,465, filed on Sep. 7, 2018.
Claims priority of provisional application 62/728,457, filed on Sep. 7, 2018.
Prior Publication US 2021/0355088 A1, Nov. 18, 2021
Int. Cl.
C07D 239/47
(2006.01);
C07D 401/12
(2006.01)
CPC
C07D 239/47
(2013.01) [
C07D 401/12
(2013.01)]
8 Claims
1. A compound selected from:
or a salt thereof.