CPC C07D 413/14 (2013.01) [A61P 35/02 (2018.01); A61K 9/0019 (2013.01)] | 12 Claims |
1. A compound of formula (I) or a salt thereof:
wherein
n is 0, 1, 2, 3, or 4;
m is 0, 1, 2, 3, or 4;
each of R1, R2, R3, R4, and R5, independently, is H, C1-C10 alkyl, C2-C10 alkenyl, C2-C10 alkynyl, C3-C20 cycloalkyl, C3-C20 cycloalkenyl, C1-C20 heterocycloalkyl, C1-C20 heterocycloalkenyl, aryl, heteroaryl, halo, ORa, SRa, COORa, OC(O)Ra, C(O)Ra, C(O)NRaRb, S(O)2NRaRb, or NRaRb;
each of R6, independently, is C1-C10 alkyl, C2-C10 alkenyl, C2-C10 alkynyl, C3-C20 cycloalkyl, C3-C20 cycloalkenyl, C1-C20 heterocycloalkyl, C1-C20 heterocycloalkenyl, aryl, heteroaryl, halo, ORa, SRa, COORa, OC(O)Ra, C(O)Ra, C(O)NRaRb, S(O)2NRaRb, or NRaRb;
each of R7, independently, is C1-C10 alkyl, C2-C10 alkenyl, C2-C10 alkynyl, C3-C20 cycloalkyl, C3-C20 cycloalkenyl, C1-C20 heterocycloalkyl, C1-C20 heterocycloalkenyl, aryl, heteroaryl, halo, ORa, SRa, COORa, OC(O)Ra, C(O)Ra, C(O)NRaRb, S(O)2NRaRb, or NRaRb;
each Ra, independently, is H, C1-C10 alkyl, C2-C10 alkenyl, C2-C10 alkynyl, C3-C20 cycloalkyl, C3-C20 cycloalkenyl, C1-C20 heterocycloalkyl, C1-C20 heterocycloalkenyl, aryl, or heteroaryl; and
each Rb, independently, is H, C1-C10 alkyl, C2-C10 alkenyl, C2-C10 alkynyl, C3-C20 cycloalkyl, C3-C20 cycloalkenyl, C1-C20 heterocycloalkyl, C1-C20 heterocycloalkenyl, aryl, or heteroaryl.
|