CPC C07J 1/0011 (2013.01) [A61K 9/0019 (2013.01); A61K 9/19 (2013.01); A61K 31/5685 (2013.01); A61K 47/34 (2013.01); A61K 47/38 (2013.01); A61P 1/00 (2018.01); A61P 3/10 (2018.01); A61P 11/06 (2018.01); A61P 31/06 (2018.01); A61P 35/00 (2018.01); A61P 37/06 (2018.01)] | 20 Claims |
1. A composition, comprising
at least 30% w/w water based on total weight of the composition, and
a compound of Formula I:
wherein n is 0 to 4;
the solvate is H2O, C1-4—OH, C1-4—OH, C1-4—COOH, C1-4—COOC1-4, tetrahydrofuran, 1,4-dioxane, (CH3)2O, (C2H5)2O, HC(O)N(CH3)2, (CH3)2SO, or a combination thereof;
X is F, Cl, Br, or I;
R is a protecting group,
wherein the compound is in form of particles stabilized as an aqueous suspension in the water.
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